Opioids

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Study Tools For Opioids

Pain Management (Cheatsheet)
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Outline

Overview

      I.         Overview

A.    Derivative from the opium poppy plant

B.    Include legal (medical) and non-legal (illicit) substances

C.     Goal: Pain-relief

     II.         Mechanism of Action

A.    Mainly, inhibits CNS receptors

1.     Receptors blocked = pain receptors blocked

   III.         Types

A.    Heroin

B.    Codeine

C.     Morphine

D.    Hydrocodone

E.     Hydromorphone

F.     Meperidine

G.    Oxycodone

I.      Opium

   IV.         Indications

A.    Pain relief

B.    Reduce cough

C.    Induce anesthesia

    V.         Side Effects

A.    CNS

1.     Diuresis

2.     Miosis

3.     Convulsions

4.     Nausea

5.     Vomiting

6.     Respiratory depression

B.    Non-CNS (d/t histamine release)

1.     Vasodilation = hypotension

2.     Colon spasms = constipation

3.     Increased ureter contractions = Decreased urine flow

4.     Dilation of cutaneous blood vessels = Flushing

   VI.         Reversal Agents

A.    Overview

1.     Block opioids receptors

a.     Respiratory depression

B.    Naltrexone

C.     Naloxone

 VII.         Withdrawal

A.    Nausea / Vomiting

B.    Confusion

C.     Muscle aches

D.    Rhinorrhea

E.     Sweating

F.     Diarrhea

G.    Fever / Chills

H.    Insomnia

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Transcript

Welcome back and today we are going to talk about opioids.

Opioids are derived from the opium poppy plant, and include legal (pharmaceuticals) and non-legal (illicit) substances. The primary goal is pain relief.

The main mechanism of action is it’s inhibition of CNS receptors. When those are blocked, pain receptors are blocked. Again, all comes back to pain relief.

There are many types of opioids. You have probably already heard of heroin and opium. These are the non-pharmaceutical types. All the others in this list are manufactured. Many people are prescribed pain medications listed here, they are highly addictive and some are in the news for the opioid epidemic.

The main indication for opioids is pain relief. Others include cough suppression and anesthesia.

Now opioids are two side effect categories, CNS and non-CNS. Pain relief can cause pinpoint pupils (an autonomic system reaction), convulsions, nausea, vomiting and respiratory depression (d/t decrease respiratory responses = slower to no respirations). Non-CNS effects are due to overall  histamine release and include hypotension, constipation, decreased urine low and flushing.

As we are in the opioid epidemic, let’s review reversal agents. Now these two block opioids receptors. So, if you patient has overdosed – this drug is given to reverse the lethal effects – usually related to respiratory depression. Due to the current opioid epidemic many first responders and even police now carry naloxone with them d/t it’s being a common occurrence. These patients are often brought to the ED, placed on mechanical ventilation to support their decrease respiratory drive and started on a narcan drip until the drug is out of their system. The goal is proper oxygenation and ventilation while the drug works itself out of their body.

Now with opiods comes addiction and dependence. These patients come in with N/V/D, confusion, aches, sweating, fever, chills and insomnia. They even can present as agitated or aggressive depending on their stage of withdrawal. Safety is an important element when managing opioid withdrawal patients.

Priority nursing concepts for a patent received opioids include comfort and pharmacology.

Alright let’s recap, there are various types of opiods, some illicit and some pharmaceutical. Usually once a person isn’t allowed anymore pharmaceutical meds, they move right to illicit drugs to support their habit if they are addicted (sadly). Indications for opioids include pain relief, cough reduction and anesthesia. Side effects are CNS or non-CNS base – # 1 being respiratory depression. Reversal agents are used if someone is found to be in respiratory distress and drugs like Narcan block opiods receptors. Lastly, withdrawal can present with a number of symptoms but make sure you are safe and know that management focus on symptoms (be antiemetics, tylenol, hydration, etc).

You know now the important details regarding opiods. Now, go out and be your best self today and as always, Happy Nursing!

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Pharmacololgy/Dosage Calc

Concepts Covered:

  • Upper GI Disorders
  • Anxiety Disorders
  • Depressive Disorders
  • Medication Administration
  • Disorders of the Posterior Pituitary Gland
  • Respiratory Disorders
  • Female Reproductive Disorders
  • Neurologic and Cognitive Disorders
  • Shock
  • Cardiac Disorders
  • Cardiovascular Disorders
  • Urinary Disorders
  • Pregnancy Risks
  • Disorders of Pancreas
  • Liver & Gallbladder Disorders
  • Hematologic Disorders
  • Substance Abuse Disorders
  • Nervous System
  • Personality Disorders
  • Dosage Calculations
  • Urinary System
  • Learning Pharmacology
  • Immunological Disorders
  • Test Taking Strategies
  • Prefixes
  • Suffixes
  • Labor Complications
  • Intraoperative Nursing
  • Prenatal Concepts
  • Postpartum Complications
  • Bipolar Disorders
  • Psychotic Disorders
  • Postoperative Nursing
  • Central Nervous System Disorders – Brain
  • Peripheral Nervous System Disorders
  • Vascular Disorders
  • Lower GI Disorders
  • Acute & Chronic Renal Disorders
  • Disorders of the Thyroid & Parathyroid Glands
  • Gastrointestinal Disorders
  • Neurological
  • Noninfectious Respiratory Disorder
  • EENT Disorders
  • Male Reproductive Disorders
  • Infectious Respiratory Disorder
  • Microbiology
  • Emergency Care of the Cardiac Patient
  • Musculoskeletal Trauma
  • Integumentary Disorders
  • Disorders of the Adrenal Gland
  • Sexually Transmitted Infections
  • Adult
  • Concepts of Pharmacology

Study Plan Lessons

Proton Pump Inhibitors
SSRIs
TCAs
Vasopressin
Anti-Infective – Penicillins and Cephalosporins
Metronidazole (Flagyl) Nursing Considerations
Ciprofloxacin (Cipro) Nursing Considerations
Vancomycin (Vancocin) Nursing Considerations
Nitro Compounds
NSAIDs
Parasympatholytics (Anticholinergics) Nursing Considerations
Hydralazine (Apresoline) Nursing Considerations
Insulin
Magnesium Sulfate
MAOIs
Histamine 1 Receptor Blockers
Histamine 2 Receptor Blockers
Histamine 2 Receptor Blockers
HMG-CoA Reductase Inhibitors (Statins)
Corticosteroids
Diuretics (Loop, Potassium Sparing, Thiazide, Furosemide/Lasix)
Epoetin Alfa
Benzodiazepines
Calcium Channel Blockers
Parasympathomimetics (Cholinergics) Nursing Considerations
Cardiac Glycosides
Autonomic Nervous System (ANS)
Sympathomimetics (Alpha (Clonodine) & Beta (Albuterol) Agonists)
ACE (angiotensin-converting enzyme) Inhibitors
Angiotensin Receptor Blockers
Atypical Antipsychotics
Injectable Medications
IV Infusions (Solutions)
Complex Calculations (Dosage Calculations/Med Math)
Renin Angiotensin Aldosterone System
Basics of Calculations
Dimensional Analysis Nursing (Dosage Calculations/Med Math)
Oral Medications
The SOCK Method – S
The SOCK Method – O
The SOCK Method – C
The SOCK Method – K
Essential NCLEX Meds by Class
6 Rights of Medication Administration
The SOCK Method – Overview
12 Points to Answering Pharmacology Questions
54 Common Medication Prefixes and Suffixes
Betamethasone and Dexamethasone in Pregnancy
Sedatives-Hypnotics
Opioid Analgesics in Pregnancy
Meds for Postpartum Hemorrhage (PPH)
Uterine Stimulants (Oxytocin, Pitocin) Nursing Considerations
Tocolytics
Mood Stabilizers
Antipsychotics
Antianxiety Meds
Magnesium Sulfate (MgSO4) Nursing Considerations
Meperidine (Demerol) Nursing Considerations
Morphine (MS Contin) Nursing Considerations
Phenobarbital (Luminal) Nursing Considerations
Pentobarbital (Nembutal) Nursing Considerations
Neostigmine (Prostigmin) Nursing Considerations
Meropenem (Merrem) Nursing Considerations
Selegiline (Eldepyrl) Nursing Considerations
Norepinephrine (Levophed) Nursing Considerations
Vasopressin (Pitressin) Nursing Considerations
Nitroglycerin (Nitrostat) Nursing Considerations
Nitroprusside (Nitropress) Nursing Considerations
Hydralazine (Apresoline) Nursing Considerations
Methylprednisolone (Solu-Medrol) Nursing Considerations
Fluticasone (Flonase) Nursing Considerations
Propofol (Diprivan) Nursing Considerations
Phenazopyridine (Pyridium) Nursing Considerations
Iodine Nursing Considerations
Sympatholytics (Alpha & Beta Blockers)
Oxycodone (OxyContin) Nursing Considerations
Nalbuphine (Nubain) Nursing Considerations
Methadone (Methadose) Nursing Considerations
Hydromorphone (Dilaudid) Nursing Considerations
Butorphanol (Stadol) Nursing Considerations
Oxytocin (Pitocin) Nursing Considerations
Hydrocodone-Acetaminophen (Vicodin, Lortab) Nursing Considerations
Methylergonovine (Methergine) Nursing Considerations
Terbutaline (Brethine) Nursing Considerations
Naproxen (Aleve) Nursing Considerations
Ketorolac (Toradol) Nursing Considerations
Indomethacin (Indocin) Nursing Considerations
Calcium Acetate (PhosLo) Nursing Considerations
Lithium (Lithonate) Nursing Considerations
Propylthiouracil (PTU) Nursing Considerations
Glucagon (GlucaGen) Nursing Considerations
Pantoprazole (Protonix) Nursing Considerations
Omeprazole (Prilosec) Nursing Considerations
Sucralfate (Carafate) Nursing Considerations
Pancrelipase (Pancreaze) Nursing Considerations
Ondansetron (Zofran) Nursing Considerations
Metoclopramide (Reglan) Nursing Considerations
Loperamide (Imodium) Nursing Considerations
Lactulose (Generlac) Nursing Considerations
Spironolactone (Aldactone) Nursing Considerations
Mannitol (Osmitrol) Nursing Considerations
Hydrochlorothiazide (Hydrodiuril) Nursing Considerations
Salmeterol (Serevent) Nursing Considerations
Montelukast (Singulair) Nursing Considerations
Guaifenesin (Mucinex) Nursing Considerations
Dopamine (Inotropin) Nursing Considerations
Olanzapine (Zyprexa) Nursing Considerations
Methylphenidate (Concerta) Nursing Considerations
Quetiapine (Seroquel) Nursing Considerations
Haloperidol (Haldol) Nursing Considerations
Tetracycline (Panmycin) Nursing Considerations
Trimethoprim-Sulfamethoxazole (Bactrim) Nursing Considerations
Amoxicillin (Amoxil) Nursing Considerations
Vancomycin (Vancocin) Nursing Considerations
Levofloxacin (Levaquin) Nursing Considerations
Rifampin (Rifadin) Nursing Considerations
Nystatin (Mycostatin) Nursing Considerations
Isoniazid (Niazid) Nursing Considerations
Metronidazole (Flagyl) Nursing Considerations
Verapamil (Calan) Nursing Considerations
Nifedipine (Procardia) Nursing Considerations
Losartan (Cozaar) Nursing Considerations
Lisinopril (Prinivil) Nursing Considerations
Propranolol (Inderal) Nursing Considerations
Metoprolol (Toprol XL) Nursing Considerations
Ranitidine (Zantac) Nursing Considerations
Promethazine (Phenergan) Nursing Considerations
Insulin – Long Acting (Lantus) Nursing Considerations
Insulin – Mixtures (70/30)
Insulin – Intermediate Acting (NPH) Nursing Considerations
Insulin – Short Acting (Regular) Nursing Considerations
Insulin – Rapid Acting (Novolog, Humalog) Nursing Considerations
Metformin (Glucophage) Nursing Considerations
Sertraline (Zoloft) Nursing Considerations
Paroxetine (Paxil) Nursing Considerations
Phenytoin (Dilantin) Nursing Considerations
Heparin (Hep-Lock) Nursing Considerations
Lamotrigine (Lamictal) Nursing Considerations
Levetiracetam (Keppra) Nursing Considerations
Streptokinase (Streptase) Nursing Considerations
Procainamide (Pronestyl) Nursing Considerations
Warfarin (Coumadin) Nursing Considerations
Midazolam (Versed) Nursing Considerations
Lorazepam (Ativan) Nursing Considerations
Opioids
Coumarins
Glipizide (Glucotrol) Nursing Considerations
Gentamicin (Garamycin) Nursing Considerations
Furosemide (Lasix) Nursing Considerations
Gabapentin (Neurontin) Nursing Considerations
Ferrous Sulfate (Iron) Nursing Considerations
Fentanyl (Duragesic) Nursing Considerations
Fluoxetine (Prozac) Nursing Considerations
Famotidine (Pepcid) Nursing Considerations
Escitalopram (Lexapro) Nursing Considerations
Erythromycin (Erythrocin) Nursing Considerations
Epoetin (Epogen) Nursing Considerations
Epinephrine (EpiPen) Nursing Considerations
Enoxaparin (Lovenox) Nursing Considerations
Enalapril (Vasotec) Nursing Considerations
Dobutamine (Dobutrex) Nursing Considerations
Divalproex (Depakote) Nursing Considerations
Diphenoxylate-Atropine (Lomotil) Nursing Considerations
Diphenhydramine (Benadryl) Nursing Considerations
Diltiazem (Cardizem) Nursing Considerations
Digoxin (Lanoxin) Nursing Considerations
Diazepam (Valium) Nursing Considerations
Dexamethasone (Decadron) Nursing Considerations
Cyclosporine (Sandimmune) Nursing Considerations
Cortisone (Cortone) Nursing Considerations
Codeine (Paveral) Nursing Considerations
Clopidogrel (Plavix) Nursing Considerations
Clindamycin (Cleocin) Nursing Considerations
Ciprofloxacin (Cipro) Nursing Considerations
Cimetidine (Tagamet) Nursing Considerations
Chlorpromazine (Thorazine) Nursing Considerations
Cefdinir (Omnicef) Nursing Considerations
Cephalexin (Keflex) Nursing Considerations
Celecoxib (Celebrex) Nursing Considerations
Cefaclor (Ceclor) Nursing Considerations
Carbidopa-Levodopa (Sinemet) Nursing Considerations
Carbamazepine (Tegretol) Nursing Considerations
Captopril (Capoten) Nursing Considerations
Calcium Carbonate (Tums) Nursing Considerations
Anti-Platelet Aggregate
Buspirone (Buspar) Nursing Considerations
Bupropion (Wellbutrin) Nursing Considerations
Bismuth Subsalicylate (Pepto-Bismol) Nursing Considerations
Bisacodyl (Dulcolax) Nursing Considerations
Benztropine (Cogentin) Nursing Considerations
Azithromycin (Zithromax) Nursing Considerations
Atropine (Atropen) Nursing Considerations
Atorvastatin (Lipitor) Nursing Considerations
Atenolol (Tenormin) Nursing Considerations
ASA (Aspirin) Nursing Considerations
Ampicillin (Omnipen) Nursing Considerations
Amlodipine (Norvasc) Nursing Considerations
Amitriptyline (Elavil) Nursing Considerations
Amiodarone (Pacerone) Nursing Considerations
Alteplase (tPA, Activase) Nursing Considerations
Alprazolam (Xanax) Nursing Considerations
Alendronate (Fosamax) Nursing Considerations
Albuterol (Ventolin) Nursing Considerations
Adenosine (Adenocard) Nursing Considerations
Acyclovir (Zovirax) Nursing Considerations
Anti-Infective – Antivirals
Acetaminophen (Tylenol) Nursing Considerations
Anti-Infective – Antifungals
Anti-Infective – Tetracyclines
Anti-Infective – Sulfonamides
Anti-Infective – Fluoroquinolones
Anti-Infective – Macrolides
Anti-Infective – Carbapenems
Anti-Infective – Aminoglycosides
Parasympathomimetics (Cholinergics) Nursing Considerations
Sympathomimetics (Alpha (Clonodine) & Beta (Albuterol) Agonists)
ACLS (Advanced cardiac life support) Drugs
The SOCK Method – Overview
The SOCK Method – O
The SOCK Method – C
The SOCK Method – K
The SOCK Method – S
Complex Calculations (Dosage Calculations/Med Math)
IV Infusions (Solutions)
Injectable Medications
Oral Medications
Dimensional Analysis Nursing (Dosage Calculations/Med Math)
Basics of Calculations
Pharmacokinetics
Pharmacodynamics
NG Tube Medication Administration
Disease Specific Medications
Vasopressin
TCAs
SSRIs
Proton Pump Inhibitors
Anti-Infective – Penicillins and Cephalosporins
Parasympatholytics (Anticholinergics) Nursing Considerations
NSAIDs
Nitro Compounds
MAOIs
Magnesium Sulfate
Insulin
HMG-CoA Reductase Inhibitors (Statins)
Hydralazine
Histamine 2 Receptor Blockers
Histamine 1 Receptor Blockers
Epoetin Alfa
Diuretics (Loop, Potassium Sparing, Thiazide, Furosemide/Lasix)
Corticosteroids
Cardiac Glycosides
Calcium Channel Blockers
Benzodiazepines
Autonomic Nervous System (ANS)
Atypical Antipsychotics
Angiotensin Receptor Blockers
ACE (angiotensin-converting enzyme) Inhibitors
Renin Angiotensin Aldosterone System
6 Rights of Medication Administration
Essential NCLEX Meds by Class
Therapeutic Drug Levels (Digoxin, Lithium, Theophylline, Phenytoin)
54 Common Medication Prefixes and Suffixes
12 Points to Answering Pharmacology Questions
Pharmacology Course Introduction